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NOVEL DERIVATIVES OF 3-HYDROXYPYRIDINE-2-CARBOXYLIC ACID, METHOD OF OBTAINING THEM, PHARMACEUTIC AGENT, APPLICATION OF SUCH DERIVATIVES AND METHOD OF OBTAINING SUCH PHARMACEUTIC AGENT
NOVEL DERIVATIVES OF 3-HYDROXYPYRIDINE-2-CARBOXYLIC ACID, METHOD OF OBTAINING THEM, PHARMACEUTIC AGENT, APPLICATION OF SUCH DERIVATIVES AND METHOD OF OBTAINING SUCH PHARMACEUTIC AGENT
N-(Esterified carboxyalkyl)-3-hydroxypyridine-2-carboxamide derivatives of formula (I) and their salts, excluding 3-Hydroxypyridine-2-carboxylic acid (glycyl ethyl ester)-amide (I'), are new. A = CH2 or CHMe; G = organic residue such that (I) is a pro-drug. Also claimed is use of (I), including (I'), as given below (see '
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机译:式(I)的N-(酯化的羧烷基)-3-羟基吡啶-2-羧酰胺衍生物及其盐,除了3-羟基吡啶-2-羧酸(缩水甘油基乙基酯)-酰胺(I'),是新的。 A = CH2或CHMe; G =有机残基,使得(I)为前药。还要求保护(I)的使用,包括(I'),如下所示(请参阅“
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