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Oxazolidinone antibacterial agents having a six-membered heteroaromatic ring.
Oxazolidinone antibacterial agents having a six-membered heteroaromatic ring.
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机译:具有六元杂芳族环的恶唑烷酮抗菌剂。
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摘要
This invention provides a novel oxazolidinone derivative represented by Formula I or pharmaceutical acceptable salts thereof: IMAGE I wherein R1 is substituted or unsubstituted 2-pyrimidinyl, 4-pyrimidinyl, or 3-pyridazinyl; X is hydrogen or fluoro; R3 is C1-4 alkyl, C1-4 alkoxy, C3-6 cycloalkyl or C1-4 alkylamino or dialkylamino. The compounds are useful antimicrobial agents.
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机译:本发明提供了一种由式Ⅰ表示的新颖的恶唑烷酮衍生物或其药学上可接受的盐:式I:其中R 1是取代或未取代的2-嘧啶基,4-嘧啶基或3-吡啶嗪基; X是氢或氟; R 3是C 1-4烷基,C 1-4烷氧基,C 3-6环烷基或C 1-4烷基氨基或二烷基氨基。该化合物是有用的抗微生物剂。
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