DERIVATIVES OF CIS-EPOXIDES, USABLE AS IRREVERSIBLE INHIBITORS OF HIV PROTEASE, AND PROCEDURES AND INTERMEDIARIES FOR THEIR PREPARATION.

摘要

THE PRESENT INVENTION REFERS TO COMPOUNDS OF CIS-EPOXIDES REPRESENTED BY FORMULA (I-1), (I-2) OR (I-3) THAT ARE USEFUL FOR THE TREATMENT OR PREVENTION OF DISEASES CAUSED BY HIV INFECTION: WHERE: A, B, D, E, R1, R10, R11, K, G, Q, R AND J HAVE THE MEANINGS DEFINED IN THE SPECIFICATION.