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SUBSTITUTED AMINO COMPOUNDS, THEIR PREPARATION AND USE AS INHIBITING SUBSTANCES OF THE THROMBOCYTE AGGREGATION.

机译:取代的氨基酸化合物,它们的制备和用作血栓凝聚素的抑制物质。

摘要

THE PRESENT INVENTION REFERS TO COMPOUNDS OF THE GENERAL FORMULA (I): R {SUP.1} - (A) {SUB.A} - (B) {B} - (D) {SUB.C} (CH {SUB .2}) {SUB.M} - N (R {SUP.2} - (CH {SUB.2}) {SUB.N} - R {SUP.3}, WHERE A, B, D, R {SUP .1} UNTIL R {SUP.3}, AS WELL AS A, B, C, MYN ARE DEFINED ACCORDING TO THE MEANING GIVEN IN THE DESCRIPTION, PROCESS FOR THEIR PREPARATION AND THEIR USE AS INHIBITORS OF THROMBOCIT AGGREGATION, OF CARCINOMA CELL METASTASIS AS WELL AS THE OSTEOPLASTIC UNION ON THE SURFACE OF THE BONES.
机译:本发明涉及通式(I)的化合物:R {SUP.1}-(A){SUB.A}-(B){B}-(D){SUB.C}(CH {SUB。 2}){SUB.M}-N(R {SUP.2}-(CH {SUB.2}){SUB.N}-R {SUP.3},其中A,B,D,R {SUP。 1}直到R {SUP.3}以及A,B,C,MYN的定义均已根据以下说明进行了定义:制备,将其制备过程以及将其用作血栓聚集抑制剂以及癌细胞转移的抑制剂作为骨骼表面上的骨质疏松联盟。

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