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COMPOUNDS EXHIBITING ANTIHYPERTENSIVE, CARDIOPROTECTIVE, ANTI-ISCHAEMIC AND ANTI-LYPOLYTIC PROPERTIES

机译:具有抗高血压,抗心脏病,抗缺血和抗溶聚性的化合物

摘要

This invention relates to adenosine derivatives and analogues which possess biological activity and are useful as anti-hypertensive, cardioprotective, anti-ischemic, and antilipolytic agents, to pharmaceutical compositions including such compounds, and to their use in treating hypertension, myocardial ischemia, ameliorating ischemic injury and myocardial infarct size consequent to myocardial ischemia, and treating hyperlipidemia and hypercholesterolemia, and to methods and intermediates used in the preparation of such compounds.
机译:本发明涉及具有生物活性并可用作抗高血压药,心脏保护药,抗缺血药和抗脂解药的腺苷衍生物和类似物,涉及包括这类化合物的药物组合物,及其在治疗高血压,心肌缺血,改善缺血性中的用途。心肌缺血,治疗高脂血症和高胆固醇血症以及制备此类化合物所用的方法和中间体所导致的损伤和心肌梗塞的大小。

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