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COMPOUNDS EXHIBITING ANTIHYPERTENSIVE, CARDIOPROTECTIVE, ANTI-ISCHAEMIC AND ANTI-LYPOLYTIC PROPERTIES

机译:具有抗高血压,抗心脏病,抗缺血和抗溶聚性的化合物

摘要

This invention relates to adenosine derivatives of the general formula I, their use for treating cardiovascular diseases, for ameliorating ischemic injury or reducing myocardial infarct size consequent to myocardial ischemia, further for reducing lipid levels, triglyceride levels, or cholesterol levels in a mammal, and for treating a cardiovascular disease bearing traces of hypertension or myocardial ischemia, reducing myocardial infarct size consequent to myocardial ischemia or for reducing lipid levels, triglyceride levels, or cholesterol levels in mammals. Disclosed is also the use of these derivatives for preparing a medicament used for treating the aforementioned diseases, as well as process for preparing these compounds.
机译:本发明涉及通式I的腺苷衍生物,其用于治疗心血管疾病,改善缺血性损伤或减少由心肌缺血导致的心肌梗塞大小,进一步降低哺乳动物中的脂质水平,甘油三酸酯水平或胆固醇水平的用途,以及用于治疗患有高血压或心肌缺血痕迹的心血管疾病,减少因心肌缺血而导致的心肌梗塞面积或降低哺乳动物的脂质水平,甘油三酸酯水平或胆固醇水平。还公开了这些衍生物在制备用于治疗上述疾病的药物中的用途,以及制备这些化合物的方法。

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