首页> 外国专利> (-)-CIS-4-AMINO-5-FLUORO-1-(2-HYDROXYMETHYL-1,3-OXATHIOLAN- -5-YL)-(1H)-PYRIMIDIN-2-ONE, A MIXTURE AND PHARMACEUTICAL COMPOSITION CONTAINING THEREOF, A COMPOUND OR MIXTURE FOR USE IN THERAPY AND FOR THE PREPARATION OF MATERIA MEDICA

(-)-CIS-4-AMINO-5-FLUORO-1-(2-HYDROXYMETHYL-1,3-OXATHIOLAN- -5-YL)-(1H)-PYRIMIDIN-2-ONE, A MIXTURE AND PHARMACEUTICAL COMPOSITION CONTAINING THEREOF, A COMPOUND OR MIXTURE FOR USE IN THERAPY AND FOR THE PREPARATION OF MATERIA MEDICA

机译:(-)-CIS-4-AMINO-5-FLUORO-1-(2-羟基甲基-1,3-氧杂环丁烷--5-基)-(1H)-吡咯烷酮-2-一,含有其的混合物和药物组合物,用于治疗和制备药物的化合物或混合物

摘要

Disclosed is a (-)-cis-4-amino-5-fluoro-1-(2-hydroxymethyl- -1,3-oxathiolan-5-yl)-(1H)-pyrimidin-2-one and its pharmaceutically acceptable salts, esters or salts of said esters as well as their pharmaceutical utilisation in the preparation of formulations used in the treatment of viral infections. There is also disclosed a pharmaceutical composition which contains one of said compounds as its active substance.
机译:公开了一种(-)-顺-4-氨基-5-氟-1-(2-羟甲基-1,3-氧杂硫杂环戊-5-基)-(1H)-嘧啶-2-酮及其药学上可接受的盐,所述酯的酯或盐以及它们在制备用于治疗病毒感染的制剂中的药物用途。还公开了包含所述化合物之一作为其活性物质的药物组合物。

著录项

  • 公开/公告号SK280131B6

    专利类型

  • 公开/公告日1999-08-06

    原文格式PDF

  • 申请/专利权人 BIOCHEM PHARMA INC.;

    申请/专利号SK19940000104

  • 发明设计人 DIONNE GERVAIS;

    申请日1992-07-24

  • 分类号C07D411/04;A61K31/505;

  • 国家 SK

  • 入库时间 2022-08-22 02:26:10

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