首页> 外国专利> DERIVATIVES OF THE ASPARTIC ACID OR ITS APPROVALS AND ITS APPLICATION IN THE TREATMENT OF DISORDERS OF THE CENTRAL NERVOUS SYSTEM.

DERIVATIVES OF THE ASPARTIC ACID OR ITS APPROVALS AND ITS APPLICATION IN THE TREATMENT OF DISORDERS OF THE CENTRAL NERVOUS SYSTEM.

机译:丙二酸的衍生物或其批准及其在治疗中枢神经系统疾病中的应用。

摘要

A PHARMACEUTICAL COMPOUND OF THE FORMULA _ (I) IN WHICH M IS 0, 1 O 2, NYQ EACH ONE 0 O 5 AND P IS 0 O 1, X IS -CO2H OR TETRAZOLYL, AND IS -CH = CH-, YZ IS (I) PHENYL, NAPHTHYL OR TENYL, OPTIONALLY SUBSTITUTED TENYL BEING SAID (II), -CHR1R2 WHERE R1 AND R2 ARE EACH PHENYL, NAPHTHYL OR TENYL WHICH IS SAYING FENYL, NAFTILE AND TENILE, REPLACED (R1) AND R2 EACH PHENYL NAPHTHYL OR TENYL, WHICH IS OPENLY SUBSTITUTED PHENYL, NAPHTHYL AND TENYL, OR (IV) WHERE R IS 0 1 TO 3 AND THE PHENYL RINGS ARE OPTIONALLY REPLACED; ALWAYS WHEN Z IS FENYL YM IS 1; AND SALTS AND ESTERS OF THESE.
机译:M为0、1 O 2,NYQ分别为0 O 5和P为0 O 1时,X为-CO2H或四唑,且-CH = CH-,YZ为(I)苯,萘基或烯丙基,可选被取代的烯丙基(II),-CHR1R2(其中R1和R2分别表示苯基,萘基和苯甲酰基,苯基和萘基),(R1或R2)苯甲基,其中的苯甲酸酯是萘,萘基和苯甲基,或者是(IV)R为0 1至3且可以选择性取代苯环的化合物;当Z为FENYL YM始终为1时;和这些盐和酯。

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