首页> 外国专利> LITHIUM SALTS OF (I'R,5'R)-3'-AZA-3'-(AZIDONAPHTHALINE-1- SULFAMIDO)-1'-(6-AMINOPURINYL-9)-3'-DEOXYHEXOPIRANOZYL- 6'-DI-OR TRIPHOSPHATES AS SPESIFIC PHOTOACTIVATED IRREVERSIBLE INHIBITORS OF Na, K-ADENOSINE TRIPHOSPHATASE

LITHIUM SALTS OF (I'R,5'R)-3'-AZA-3'-(AZIDONAPHTHALINE-1- SULFAMIDO)-1'-(6-AMINOPURINYL-9)-3'-DEOXYHEXOPIRANOZYL- 6'-DI-OR TRIPHOSPHATES AS SPESIFIC PHOTOACTIVATED IRREVERSIBLE INHIBITORS OF Na, K-ADENOSINE TRIPHOSPHATASE

机译:(I'R,5'R)-3'-AZA-3'-(叠氮萘基-1-硫代酰胺)-1'-(6-氨基壬基-9)-3'-脱氧己基吡咯烷基-6'-DI-的锂盐或三磷酸酯作为Na,K-腺苷三磷酸酯酶的特定的光活化不可逆抑制剂

摘要

FIELD: biochemistry. SUBSTANCE: lithium salts of (1'R, 5'R)-3'-aza-3'-azidonaphthalene-1- sulfamino-1'-(6-amino-purinyl-9)-3'-deoxyhexopyranozyl-6- di-or triphosphates of general formula I: R1=N3,R2=H or R1=H and R2=N3 wherein n is 2 or 3, are useful for specific inhibition of Na, K-adenonosine triphosphatase. EFFECT: improved properties of the title compounds. 4 ex, 1 tbl
机译:领域:生物化学。物质:(1'R,5'R)-3'-氮杂-3'-叠氮萘-1-磺氨基-1'-(6-氨基嘌呤基-9)-3'-脱氧己吡喃并基-6-二锂盐-或通式I的三磷酸酯:R 1 = N 3 ,R 2 = H或R 1 = H和R 2 = N 3 ,其中n为2或3,可用于特异性抑制Na,K-腺苷三磷酸酶。效果:改善了标题化合物的性质。 4桶1桶

著录项

相似文献

  • 专利
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号