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TETRAHYDRO-1H-BENZAZEPINONE AND HEXAHYDRO AZEPINONE AS SELECTIVE CHOLECYSTOKININ-B RECEPTOR ANTAGONISTS
TETRAHYDRO-1H-BENZAZEPINONE AND HEXAHYDRO AZEPINONE AS SELECTIVE CHOLECYSTOKININ-B RECEPTOR ANTAGONISTS
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机译:四氢-1H-苯并ZE庚酮和六氢苯并PIN庚酮为选择性胆囊收缩素-B受体拮抗剂
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PCT No. PCT/IB94/00111 Sec. 371 Date Jan. 18, 1996 Sec. 102(e) Date Jan. 18, 1996 PCT Filed May 19, 1994 PCT Pub. No. WO95/03281 PCT Pub. Date Feb. 2, 1995This invention relates to compounds of formula (I) wherein R1, R2, R3, R4 and X are as defined in the application. These compounds are CCK-B receptor antagonists and are useful in the treatment and prevention of central nervous system and gastrointestinal disorders. IMAGE (I)
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