首页> 外国专利> NOVEL PEPTIDE, AND PLATELET AGGREGATION-INHIBITING AGENTS, BLOOD COAGUL ATION-INHIBITING AGENTS FOR EXTRACORPOREAL CIRCULATION, CELL ADHESION-INHIBITING AGENTS, TUMOR METASTASIS-INHIBITING AGENTS, AGENTS FOR PROTECTING PLATELET PREPARATIONS FOR BLOOD TRANSFUSION, PLATELET PREPARATIONS AND PLATELET PREPARATION PACKS FOR TRANSFUSION USING SAID NOVEL PEPTIDES

NOVEL PEPTIDE, AND PLATELET AGGREGATION-INHIBITING AGENTS, BLOOD COAGUL ATION-INHIBITING AGENTS FOR EXTRACORPOREAL CIRCULATION, CELL ADHESION-INHIBITING AGENTS, TUMOR METASTASIS-INHIBITING AGENTS, AGENTS FOR PROTECTING PLATELET PREPARATIONS FOR BLOOD TRANSFUSION, PLATELET PREPARATIONS AND PLATELET PREPARATION PACKS FOR TRANSFUSION USING SAID NOVEL PEPTIDES

机译:新型肽和抑制血小板凝集的试剂,用于体外循环的血凝抑制试剂,抑制细胞粘附的试剂,抑制肿瘤转移的试剂,用于制备血小板制备的试剂盒,制备血小板制备制剂的制剂新型肽

摘要

The present invention provides compounds or salts thereof, that are represented by the general formula (I): Pro-Ser-A-B-Asp-C-D,wherein A is an amino acid other than amino acids having a guanidino group at a side chain, B is an amino acid, C is an amino acid havinga hydrophobic group at a side chain and D is a hydroxy or an amino group. The compounds and salts thereof of the present invention areuseful since they have excellent platelet aggregation-inhibiting and blood coagulation-inhibiting activities and are highly safe.
机译:本发明提供由通式(I)表示的化合物或其盐:Pro-Ser-A-B-Asp-C-D,其中A是除在侧链具有胍基的氨基酸以外的氨基酸,B是氨基酸,C是具有侧链上的疏水基团,D是羟基或氨基。本发明的化合物及其盐是因为它们具有优异的抑制血小板聚集和抑制凝血的活性并且非常安全,所以它们是有用的。

著录项

  • 公开/公告号CA2168964C

    专利类型

  • 公开/公告日2000-08-22

    原文格式PDF

  • 申请/专利权人

    申请/专利号CA19942168964

  • 发明设计人 SATO YOSHIMI;HAYASHI YOSHIO;KATADA JUN;

    申请日1994-09-29

  • 分类号C07K7/06;A61K38/08;

  • 国家 CA

  • 入库时间 2022-08-22 01:53:11

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