首页> 外国专利> 6-Amino- or 6-hydrazino-sulfonyl-3-quinolinyl-phosphonic acid compounds, process for their preparation and pharmaceutical compositions containing them

6-Amino- or 6-hydrazino-sulfonyl-3-quinolinyl-phosphonic acid compounds, process for their preparation and pharmaceutical compositions containing them

机译：6-氨基或6-肼基-磺酰基-3-喹啉基-膦酸化合物，其制备方法和含有它们的药物组合物

页面导航

摘要
著录项
相似文献

摘要

Invention Patent: B "6-AMINO- OR 6-HYDRAZINO-SULFONYL-3-QUINOLINYL-PHOSPHENIC ACID COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM" D. This invention relates to compounds of formula (I): where: sym R¹ represents a halogen atom or a CF ~ 3 ~ group, sym R² represents a hydrogen atom or an alkyl or cycloalkyl group, sym R³ is as defined in the description. sym R ^ 4 ^ and R ^ 5 ^ represent a hydrogen atom or an alkyl, cycloalkyl, aryl or arylalkyl group, or a Medicines group.

机译：发明专利：“ 6-氨基-或6-肼基-磺酰基-3-喹啉基-膦酸化合物，其制备方法和含有它们的药物组合物” 。本发明涉及式（Ⅰ）化合物：其中：式中R 1代表卤原子或CF 3-基团，式中R 2代表氢原子或烷基或环烷基，式中R 3如上。在说明中定义。 <符号> R ^ 4 ^和R ^ 5 ^代表氢原子或烷基，环烷基，芳基或芳基烷基或药物基团。 展开▼

著录项

公开/公告号BR0100601A

专利类型

公开/公告日2001-09-18

原文格式PDF

申请/专利权人 ADIR ET COMPAGNIE;
展开▼

申请/专利号BR20010100601

发明设计人 ALEX CORDI;PATRICE DESOS;PIERRE LESTAGE;
展开▼

申请日2001-02-16

分类号C07D215/227;A61K31/47;A61P25/28;

国家 BR

入库时间 2022-08-22 01:26:09

相似文献

专利

外文文献

中文文献

1. 新的6－氨基或6－肼基－磺酰基3－喹啉基膦酸化合物,其制备方法及含有它们的药物组合物 [P] . 中国专利： CN1320601A . 2001-11-07

2. 新的－6－氨磺酰－3－喹啉基膦酸化合物,其制备方法及含有它们的药物组合物 [P] . 中国专利： CN1317490A . 2001-10-17

3. composition, pharmaceutical composition, effervescent dosage form, multiple unit oral oral pharmaceutical composition, extended release pharmaceutical dosage form, enteric coated pharmaceutical dosage form, stable pharmaceutical dosage form for oral administration to mammalian subjects, method for treating diseases acid-related diseases by inhibiting gastric acid secretion, method for treating a bacterial infection caused or caused by helicobacter pylori, process for preparing a compound of formula 3, process for preparing a compound of formula 5, use of a compound of formula 1 for the preparation of a medicament for treating gastric acid-related diseases by inhibiting gastric acid secretion, use of a compound of formula 1 for the preparation of a medicament for treating a bacterial infection caused or caused by helicobacter pyl or use of a compound of formula 1 for the preparation of a medicament for treating gastric acid-related diseases by inhibiting gastric acid secretion [P] . BRPI0617987A2 . 2011-08-16

机译：组合物，药物组合物，泡腾剂型，多单位口服口服药物组合物，缓释药物剂型，肠溶衣药物剂型，向哺乳动物受试者口服给药的稳定药物剂型，通过抑制胃酸治疗疾病的方法酸分泌，治疗由幽门螺杆菌引起或引起的细菌感染的方法，制备式3化合物的方法，制备式5化合物的方法，式1化合物在制备用于治疗胃的药物中的用途通过抑制胃酸分泌来治疗与酸有关的疾病，将式1的化合物用于制备用于治疗由幽门螺杆菌引起或引起的细菌感染的药物，或将式1的化合物用于制备用于治疗的药物通过抑制胃酸分泌来治疗胃酸相关疾病

4. New 6-amino- or 6-hydrazino-sulphonyl-3-quinolynyl- phosphonic acid compounds, a process for their preparation and pharmaceutical compositions containing them [P] . AU2304201A . 2001-08-23

机译：新的6-氨基或6-肼基-磺酰基-3-喹啉基-膦酸化合物，其制备方法和含有它们的药物组合物

5. 6- 6---3-- NEW 6-AMINO- OR 6-HYDRAZINO-SULPHONYL-3-QUINOLYL-PHOSPHONIC ACID COMPOUNDS A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM [P] . 韩国专利： KR20010082702A . 2001-08-30

机译： 6- 6 --- 3--新型6-氨基或6-肼基-磺酰基-3-喹啉-膦酸化合物的制备方法和包含它们的药物组合物

1. Screening Research of Pharmaceutical Compositions Based on Succinic Acid, Ascorbic Acid and Rutin [J] . Mariya Leleka, Olha Zalis＇ka, Galyna Kozyr 药剂与药理学：英文版 . 2016,第009期

2. Effects of ensiling processes and antioxidants on fatty acid concentrations and compositions in corn silages [J] . Liying Han, He Zhou 畜牧与生物技术杂志：英文版 . 2014,第002期

3. Effects of ensiling processes and antioxidants on fatty acid concentrations and compositions in corn silages [J] . Liying Han, He Zhou 畜牧与生物技术杂志(英文版) . 2014,第002期

4. Lipid Oxidation and Fatty Acid Composition in Salt-Dried Yellow Croaker (Pseudosciaena polyactis) During Processing [J] . CAI Qiuxing, WU Yanyan, LI Laihao, 中国海洋大学学报（英文版） . 2017,第005期

5. Preparation of Chiral Amino Acid Intermediatesfor Synthesis of Pharmaceutical Compounds UsingAmino Acid Dehydrogenases [C] . Ronald L. Hanson ACS symposium asymmetric synthesis and application of α-amino acids . 2009

6. Assessing Removal of Pharmaceutical Compounds in Conventional Wastewater Treatment and Ultraviolet-Peracetic Acid Advanced Oxidation Process andDevelopment of a Comprehensive Analytical Method for the Quantification of Veterinary AntimicrobialsSpanning Several LivestockIndustries [D] . Naas, Kayla. 2019

7. Echium oil with oxidative stability increased by emulsion preparation in the presence of the phenolic compound sinapic acid followed by dehydration by spray and freeze drying processes [O] . Talita A. Comunian, Luísa F. Favaro, Marcelo Thomazini, 2019

8. The Preparation of Some Amino-acids and Amino-aldehydes. III. Thermal Decomposition of Ethyl-N, N-dibenzyl-γ-aminobutyrate and Related Compounds. [O] . Shirô Morosawa 1958

1. Treatment of pharmaceutical wastewater containing recalcitrant compounds in a Fenton-coagulation process [J] . Bukuru Godefroid . 环境科学学报：英文版 . 2006,第3期

2. 具有生物活性有机磷化合物研究XXⅤα-(4,6-二氯嘧啶基氨基甲酰氧基烃基膦酸酯的合成与生物活性的研究 [C] . 贺红武 . 中国化工学会农药专业委员会第九届年会 . 1998

3. 具有生物活性的多取代-2-氨基嘧啶衍生物及其稠杂环化合物的研究（Ⅷ、Ⅸ）;Ⅷ：N'-（4,6-二取代嘧啶-2-基）-N-取代酰基硫脲的合成，晶体结构及除草活性;Ⅸ：5,7-二取代芳酰亚胺基-2H-1,2,4-噻二唑并[2,3-a]嘧啶的合成及除草活性 [A] . 王洁平 . 2003