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PHARMACEUTICAL COMPOSITION CONTAINING A CYSTEINE PROTEASE INHIBITOR FOR PROPHYLAXIS AND THERAPY OF BRAIN TISSUE IMPAIRMENT

机译:包含半胱氨酸蛋白酶抑制剂的脯氨酸类药物的药物组合物和脑组织损伤的治疗

摘要

A pharmaceutical composition for the prevention and treatment of cerebrovascular damage, wherein, as an active ingredient, wherein R1 is C1-C4 alkyl or C6-10 is optionally substituted aryl; R2 and R3 are independently hydrogen or C1-C4 alkyl, or R2 and R3 are attached to form a C3-7 ring, R4 is a lower alkyl group optionally substituted by aryl, cycloalkyl or aromatic heterocyclic group containing a pharmaceutically acceptable salt thereof. HE
机译:用于预防和治疗脑血管损伤的药物组合物,其中作为活性成分,其中R1是C1-C4烷基或C6-10是任选取代的芳基; R 2和R 3独立地是氢或C 1 -C 4烷基,或R 2和R 3连接形成C 3-7环,R 4是任选地被芳基,环烷基或含有其药学上可接受的盐的芳族杂环基取代的低级烷基。他

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