首页> 外国专利> DERIVATIVES IN THE VITAMIN D SERIES MODIFIED IN THE 20TH POSITION, A METHOD OF PREPARING SUCH DERIVATIVES, INTERMEDIATES USED IN THIS METHOD, PHARMACEUTICAL PREPARATIONS CONTAINING THE DERIVATIVES AND THEIR USE IN THE PREPARATION OF DRUGS

DERIVATIVES IN THE VITAMIN D SERIES MODIFIED IN THE 20TH POSITION, A METHOD OF PREPARING SUCH DERIVATIVES, INTERMEDIATES USED IN THIS METHOD, PHARMACEUTICAL PREPARATIONS CONTAINING THE DERIVATIVES AND THEIR USE IN THE PREPARATION OF DRUGS

机译:在20位修饰的维生素D系列中的衍生物,一种制备此类衍生物的方法,在该方法中使用的中间体,包含该衍生物的药物制剂及其在药物制备中的用途

摘要

The invention concerns vitamin D derivatives, modified in the 20th position, of general formula (I), in which Z is H, OH or C1-9 alkanoyl; X is H or both X's together mean an exocyclic methylene group; Y is H, C1-9 alkanoyl or arylcarbonyl; and meanings of other substituents are given in the claims; a method of preparing them; intermediates, pharmaceuticals containing said derivatives and their use for the preparation of medicaments.
机译:本发明涉及在通式(I)的第20位上修饰的维生素D衍生物,其中Z为H,OH或C1-9链烷酰基; X为H或两个X一起表示环外亚甲基; Y为H,C 1-9烷酰基或芳基羰基;其他取代基的含义在权利要求书中给出;一种准备方法;中间体,含有所述衍生物的药物及其在制备药物中的用途。

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