首页> 外国专利> NEW N-AMINOALQUILFLUORENOCARBOXAMIDS; A NEW CLASS OF SPECIFIC LIGANDS TO SUBTOPS OF THE DOPAMINE RECEIVER.

NEW N-AMINOALQUILFLUORENOCARBOXAMIDS; A NEW CLASS OF SPECIFIC LIGANDS TO SUBTOPS OF THE DOPAMINE RECEIVER.

机译:新的N-氨基铝氟橡胶一类新的多巴胺接收器专用子标签。

摘要

THE INVENTION REFERS TO FORMULA (I) COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS OF THE SAME. IN THIS FORMULA: G REPRESENTS A GROUP OF FORMULA (A), (B) OR (C), WHERE R A AND R B REPRESENT HYDROGEN OR ORGANIC OR INORGANIC SUBSTITUTES; A IS AN OPTIONALLY REPLACED RENT; R 1, R 2, R 3 AND R 4 REPRESENT SUBSTITUTES ORGANIC OR INORGANIC; R 5 IS HYDROGEN OR LOWER RENT; R 6 AND R 7 INDEPENDENTLY REPRESENT HYDROGEN OR LOWER RENT, OR JOINTLY FORM A CYCLE OF 5-8 MEMBERS; Z IS NITROGEN OR CARBON AND W IS ARILO OR HETEROARILO OPTIONALLY REPLACED.
机译:本发明涉及相同的化合物(I)化合物或药学上可接受的盐。在此公式中:G代表一组式(A),(B)或(C),其中R A和R B代表氢或有机或无机取代基; A是可选的租金; R 1,R 2,R 3和R 4代表有机或无机取代基; R 5是氢或更低的租金; R 6和R 7独立存在的氢或更低的租金,或共同形成5-8个成员的循环; Z是氮或碳,W是任选取代的芳基或杂芳基。

著录项

  • 公开/公告号ES2159758T3

    专利类型

  • 公开/公告日2001-10-16

    原文格式PDF

  • 申请/专利权人 NEUROGEN CORPORATION;

    申请/专利号ES19960931543T

  • 发明设计人 YUAN JUN;CHEN XI;

    申请日1996-09-12

  • 分类号C07D295/12;C07D211/70;A61K31/495;A61K31/445;

  • 国家 ES

  • 入库时间 2022-08-22 01:22:14

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