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BENZOCYCLOALKYLAMINOPYRIDINAMINES AND RELATED COMPOUNDS, A PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS

机译:苯环烷基氨基吡啶酰胺类化合物及相关化合物,其制备方法和中间体以及其用作药物

摘要

Benzocycloalkylaminopyridinamines and related compounds,a process and intermediates for their preparation and theiruse as medicamentsThere are described compounds of the formula,(see formula I)whereR is hydrogen, loweralkyl, arylloweralkyl or loweralkylearbonyl;k is 0 or 1;m is 1, 2 or 3;k+m is 2 or 3; andn is 0 or 1;which compounds are useful as topical antiinflammatory agents for thetreatmentof various dermatoses , intermediates thereof and a process fortheir preparation.
机译:苯并环烷基氨基吡啶胺和相关化合物,它们的制备及其中间体的过程和中间体用作药物描述了下式的化合物,(参见公式I)哪里R为氢,低级烷基,芳基低级烷基或低级烷基硬脂基;k为0或1;m为1、2或3;k + m是2或3;和n为0或1;哪些化合物可用作局部抗炎药治疗各种皮肤病,其中间体及其制备方法他们的准备。

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