首页> 外国专利> Preparation of Ä1s-Ä1a 2b 3b 4a(s*)ÜÜ1-(3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3h-imidazoÄ4 5-bÜpyridin-3-ylÜ-n-ethyl-2 3-dihydroxycyclopentanecarboxamide

Preparation of Ä1s-Ä1a 2b 3b 4a(s*)ÜÜ1-(3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3h-imidazoÄ4 5-bÜpyridin-3-ylÜ-n-ethyl-2 3-dihydroxycyclopentanecarboxamide

机译:Ä1s-Ä1a2b 3b 4a(s *)ÜÜ1-(3-氯-2-噻吩基)甲基Ü丙基ÜaminoÜ-3h-咪唑基Ä45-bÜpyridin-3-ylÜ-n-ethyl-23-dihydroxycyclopentaneCarboxamide的制备

摘要

This invention is directed to methods for the preparation of Ä1S-Ä1a,2b,3b,4a(S*)ÜÜ-4-Ä7-ÄÄ1-(3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3H-imidazoÄ4,5-bÜpyridi n-3-ylÜ-N-ethyl-2,3-dihydroxycyclopentanecarboxamide, methods for the preparation of intermediates thereto, and to said intermediates themselves.
机译:本发明涉及制备Ä1S-Ä1a,2b,3b,4a(S *)ÜÜ-4-Ä7-ÄÄ1-(3-氯-2-噻吩基)甲基Ü丙基ÜaminoÜ-3H-咪唑基4,5-b吡啶基的方法-3-基-N-乙基-2,3-二羟基环戊烷甲酰胺,其中间体的制备方法,以及所述中间体本身。

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