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A Pharmaceutical composition comprising a nicotine receptor agonist and a useful Analgesic for the treatment of chronic and acute pain and / or neuropathic pain and migraines

机译:包含尼古丁受体激动剂和有用的镇痛药的药物组合物,用于治疗慢性和急性疼痛和/或神经性疼痛和偏头痛

摘要

Relates to a composition useful for the treatment of chronic and acute pain, neuropathic, migrana, comprising: a) a nicotine receptor partial agonist as 9 - Bromine - 1,2,3,4,5,6 - hexahidro - 1.5 - methane - pirido [1,2-a] [1.5] diazocin ONA - 8 -, 9 - chlorine - 1 - - 1.5 - methane - hexahidro pirido [1,2-a] [1.5] diazocin - 8 - ona, among others; (b) as an Analgesic meperidine, propoxyphene,Hydrocodone, hydromorphone, morphine, tramadol, codeine, - 1 - 2 - piperidino alkanol, dextromethorphan, eliprodil, Ifenprodil,6 - methoxy - 3 - trifluoromethyl - benzo [d] isoxazole - ylmethyl) - 5 - (2 - phenyl - 3 - piperidin yl) Amine, rofecoxib, celecoxib, Nitrous Oxide Halothane, Lidocaine, ropivacaine, cloroprocaina sarapina etidocaine,,,Bupivacaine, chlordiazepoxide, diazepam, lorazepam, alprazolam, Flexeril, gabapentin, pregabalin, Salicylic Acid, Baclofen, clonidine, prednisone; (c) a vehicle
机译:涉及一种用于治疗慢性和急性疼痛,神经性,偏头痛的组合物,其包含:a)尼古丁受体部分激动剂,如9-溴-1,2,3,4,5,6-六溴-1.5-甲烷- pirido [1,2-a] [1.5]重氮ONA-8-,9-氯-1--1.5-甲烷-六羟基pirido [1,2-a] [1.5] diazocin-8-ona等; (b)作为止痛药哌替啶,丙氧芬,氢可酮,氢吗啡酮,吗啡,曲马多,可待因,-1-2-哌啶子基链烷醇,右美沙芬,依普罗地尔,Ifenprodil,6--甲氧基-3-三氟甲基-苯并[d]异恶唑-丁基甲基) -5-(2-苯基-3-哌啶基)胺,罗非昔布,塞来昔布,一氧化二氮氟烷,利多卡因,罗哌卡因,氯吡普罗那sarapina依托卡因,布比卡因,氯二氮杂卓,地西epa,劳拉西m,沙丁酸,阿普唑仑,普瑞巴林酸,巴氯芬,可乐定,泼尼松; (c)车辆

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