首页> 外国专利> Compound or a physiologically acceptable salt or solvate thereof, use thereof, pharmaceutical composition, aerosol pharmaceutical formulation, method for treating a human or animal subject with an antiinflammatory and / or allergic condition, and process for preparing a compound

Compound or a physiologically acceptable salt or solvate thereof, use thereof, pharmaceutical composition, aerosol pharmaceutical formulation, method for treating a human or animal subject with an antiinflammatory and / or allergic condition, and process for preparing a compound

机译:化合物或其生理上可接受的盐或溶剂化物,其用途,药物组合物,气雾剂药物制剂,用于治疗具有抗炎和/或过敏性疾病的人或动物受试者的方法以及制备该化合物的方法

摘要

"COMPOUND OR ITS PHYSIOLOGICALLY ACCEPTABLE SALT OR SOLVAT, USE OF THE SAME, PHARMACEUTICAL COMPOSITION, PHARMACEUTICAL FORMULATION, METHOD FOR TREATMENT OF A HUMAN OR ANIMAL INDIVIDUAL AND ANALYTIC CONDITION AND ANALYTIC CONDITION, . Provided according to the invention are compounds of formula (I) wherein R 1 - represents C 1-6 alkyl or C 1-6 haloalkyl; R2 is -C (= O) aryl or -C (= O) heteroaryl; R 3 represents hydrogen, methyl (which may be in the α or β configuration) or methylene; R4 and R5 are the same or different and each represents hydrogen or halogen; and ---- represents a single or double bond; and their salts and solvates. Processes are also provided for preparing compounds of formula (I) and use of the compounds in therapy, especially in the treatment of inflammatory and allergic conditions.
机译:“根据本发明提供的化合物或其生理上可接受的盐或溶剂,相同化合物的使用,药物成分,药物配方,人类或动物个体和分析条件及分析条件的治疗方法。其中R 1-代表C 1-6烷基或C 1-6卤代烷基; R2是-C(= O)芳基或-C(= O)杂芳基; R 3代表氢,甲基(可以在α或β中R 4和R 5相同或不同,分别代表氢或卤素;和----代表单键或双键;及其盐和溶剂化物;还提供了制备式(I)化合物的方法以及该化合物在治疗中的用途,尤其是在炎性和过敏性疾病的治疗中。

著录项

  • 公开/公告号BR0113039A

    专利类型

  • 公开/公告日2003-07-15

    原文格式PDF

  • 申请/专利权人 GLAXO GROUP LIMITED;

    申请/专利号BR20010113039

  • 申请日2001-08-03

  • 分类号C07J31/00;A61K31/58;C07J33/00;C07J71/00;C07J3/00;A61P5/44;

  • 国家 BR

  • 入库时间 2022-08-22 00:03:50

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号