首页> 外国专利> Þíól afleiður með málmpeptíðasa letjandi virkni, aðferð til framleiðslu þeirra, lyfjaefnablöndur sem innihalda slíkt efnasamband, ásamt notkun á efnasamböndunum til framleiðslu á lyfjum

Þíól afleiður með málmpeptíðasa letjandi virkni, aðferð til framleiðslu þeirra, lyfjaefnablöndur sem innihalda slíkt efnasamband, ásamt notkun á efnasamböndunum til framleiðslu á lyfjum

机译:具有金属肽酶抑制活性的硫醇衍生物,其制备方法,含有该化合物的药物制剂以及该化合物在制备医药产品中的用途

摘要

Compounds of formula (I), wherein R, R1, R2, and R3 have the meanings reported in the description, processes for their preparation and pharmaceutical compositions which contain them as active ingredients are described. The compounds of formula (I) are endowed with a mixed ACE-inhibitory and NEP-inhibitory activity and are useful in the treatment of cardiovascular diseases.
机译:描述了其中R,R1,R2和R3具有说明书中报道的含义的式(I)化合物,其制备方法和含有它们作为活性成分的药物组合物。式(I)化合物具有混合的抑制ACE和抑制NEP的活性,可用于治疗心血管疾病。

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