首页> 外国专利> DERIVATIVES OF 3,4-DIHYDROANTRACENE SUST. WITH ARYL OR HETEROARILO AND BENZO (1,2-G) -CROM-3-ENO, BENZO (1,2-G) -TIOCROM-3-ENO AND BENZO (1,2-G) -1,2-DIHYDROQUINOLINE SUST . WITH ARILO OR HETEROARILO THAT HAVE ACTIV. BIOLOGICAL AS RETINOID ANTAGONISTS OR RETINOID INVESTED AGONISTS.

DERIVATIVES OF 3,4-DIHYDROANTRACENE SUST. WITH ARYL OR HETEROARILO AND BENZO (1,2-G) -CROM-3-ENO, BENZO (1,2-G) -TIOCROM-3-ENO AND BENZO (1,2-G) -1,2-DIHYDROQUINOLINE SUST . WITH ARILO OR HETEROARILO THAT HAVE ACTIV. BIOLOGICAL AS RETINOID ANTAGONISTS OR RETINOID INVESTED AGONISTS.

机译:必须衍生出3,4-二氢蒽衍生物。与ARYL或杂芳基和苯并(1,2-G)-CROM-3-ENO,苯并(1,2-G)-TIOCROM-3-ENO和苯并(1,2-G)-1,2-二氢喹啉。与具有ACTIV的ARILO或HETEROARILO。生物作为类视黄醇拮抗剂或类视黄醇拮抗剂。

摘要

THE INVENTION REFERS TO FORMULA COMPOUNDS (1), WHERE SYMBOLS HAVE THE MEANING DEFINED IN THE DESCRIPTION. THESE COMPOUNDS PRESENT BIOLOGICAL ACTIVITY OF ANTAGONIST TYPE AND / OR REVERSE AGONIST OF THE RETINOIDS.
机译:本发明是指配方化合物(1),其中符号在说明书中定义的含义。这些化合物目前具有拮抗剂类型的生物活性和/或类视黄醇的逆向激动剂。

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