首页> 外国专利> VENLAFAXINA AND ITS ANALOGS TO INDUCE AN IMPROVEMENT OF COGNITIVE FUNCTIONS.

VENLAFAXINA AND ITS ANALOGS TO INDUCE AN IMPROVEMENT OF COGNITIVE FUNCTIONS.

机译:VENLAFAXINA及其类似物可改善认知功能。

摘要

THE INVENTION PROVIDES A COMPOUND TO MANUFACTURE A MEDICINAL PRODUCT TO INDICATE THE IMPROVEMENT OF KNOWLEDGE. THE COMPOUND IS A DERIVATIVE OF 2- (1-HYDROXICICLOALQUIL OR 1-HYDROXICICLOALQUENIL) -2 PHENYL ALKYLAMEN THAT HAS THE FORMULA (I) IN WHICH A MOLECULA OF THE FORMULA (II) IS IN WHICH THE STITCHED LINE REPRESENTS AN INSATURATION; R1 IS HYDROGEN OR RENT; R2 IS RENT; R4 IS HYDROGEN, RENT, FORMYL OR ALCANOYL; R5 AND R6 ARE, INDEPENDENTLY, HYDROGEN, HYDROXYL, RENT, ALCOXI, ALCANOILOXI, CYANO, NITRO, ALKYLMARKET, AMINO, ALQUILAMINO, DIALQUILAMINO, ALCANAMIDO, HALO, TIFLUOROMETHYLENE METHYLENE; R7 IS HYDROGEN OR RENT; AND N IS 0, 1, 2, 3 OR 4, THE PHARMACOLOGICALLY ACCEPTABLE SALTS OF THE COMPOUND ARE ALSO PRESENTED.
机译:本发明提供了一种制造医学产品以指示对知识的改进的化合物。该化合物是具有式(I)的分子式(II)的分子式(II)存在于缝线中时;该化合物的式(I)的衍生物是2-(1-羟基氯代喹啉或1-羟基羟基喹啉)-2酚烷基。 R1是氢或租金; R2已租出; R4是氢,租,甲酰基或烷酰基; R5和R6独立地是氢,氢氧根,租金,酒精,烷氧基,氰基,硝基,烷基市场,氨基酸,喹啉醇,对苯二甲胺基,烷酰胺基,卤素,三氟甲基亚甲基; R7是氢或租金;并且N为0、1、2、3或4,该化合物的药理学上可接受的盐也被提出。

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