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Treatment and prevention of the adverse effects of reactive oxygen species.

机译:治疗和预防活性氧的不利影响。

摘要

BUCILAMINE AND N-2,2-DIMETHYL-3MERCAPTOPROPIONIL) -L-CYSTEINE OR RELATED COMPOUNDS MAY BE USED TO AVOID DAMAGE TO LIVING FABRICS THAT ARE DERIVED FROM THE FORMATION OR PRESENCE OF REACTIVE OXYGEN SPECIES. THESE REAGENT SPECIES OF OXYGEN ARE FORMED WHEN THE TISSUE IS RETURNED FOR THE FIRST TIME HYPOXIC DUE TO THE INTERRUPTION OF THE BLOOD FLOW AND THEN REOXIGATES THROUGH THE RESTORATION OF THE BLOOD FLOW. IN PARTICULAR THE INVENTION REFERS TO THE ADMINISTRATION OF BUCILAMINE AND N-2,2-DIMETHYL-3MERCAPTOPROPIONIL) -L-CISTEINE BEFORE OR COINCIDING WITH THE REPERFUSION TO AVOID DAMAGE TO THE MIOCARDY THAT IS DERIVED FROM THE REACTION OF SPECIFICATION. APPLICATIONS OF THESE COMPOUNDS FOR SIMILAR CELL INJURIES RELATED TO THE ISCHEMIA OR OTHER ORGANS ARE ALSO SUBMITTED.
机译:丁二胺和N-2,2-二甲基-3巯基丙酸酯)-L-半胱氨酸或相关化合物可用于避免损害起因于活泼氧物种的形成或存在的纤维。当组织因血流中断而首次缺氧时归还氧气时,便会形成这些氧气的物种,然后通过血流恢复来补充氧气。特别地,本发明是指在再灌注之前避免对布查拉明和N-2,2-二甲基-3巯基丙酸(L-2)-L-半胱氨酸的管理,以免损害是由于规范反应而引起的。这些化合物用于缺血或其他器官相关的类似细胞损伤的应用也已提交。

著录项

  • 公开/公告号ES2185909T3

    专利类型

  • 公开/公告日2003-05-01

    原文格式PDF

  • 申请/专利号ES19970905855T

  • 发明设计人 HORWITZ LAWRENCE D.;

    申请日1997-02-07

  • 分类号A61K31/095;A61K31/16;A61K31/195;A61P9/00;

  • 国家 ES

  • 入库时间 2022-08-21 23:59:10

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