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PREPARATION OF PHARMACEUTICAL STABILITY OF NASAL ORAL OR SUB-LINGUAL APPLICATION CONTAINING DESMOPRESSIN

机译:含有去氨加压素的鼻内或舌下应用的药物稳定性的制备

摘要

A stable, nasally, orally or sublingually applicable pharmaceutical preparation for administering to patients has an aqueous solution of desmopressin as the active agent. Said solution contains an osmoticum and a buffer which maintains the pH-value in the range of 4 to 6, preferably about 5. The buffer is malic acid, preferably in the form of a racemate. Thereby an improved stability of the desmopressin content in the preparation is obtained.
机译:用于向患者给药的稳定的,经鼻,经口或舌下施用的药物制剂具有去氨加压素的水溶液作为活性剂。所述溶液包含渗透剂和保持pH值在4至6,优选约5的缓冲液。缓冲液是苹果酸,优选为外消旋体形式。由此获得了制剂中去氨加压素含量的改善的稳定性。

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