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PROCEDURE TO PREPARE NAFTIRIDONES AND INTERMEDIATES.
PROCEDURE TO PREPARE NAFTIRIDONES AND INTERMEDIATES.
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机译:制备萘啶酮和中间体的步骤。
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摘要
THE INVENTION REFERS TO A PROCEDURE FOR PREPARING A CARBOXILIC ACID OF NAFTIRIDONA AND ITS DERIVATIVES, WHICH USES THE SIDE CHAIN INTERMEDIARIES OF FORMULAS I AND IV WHERE R 1 IS BENCILO, WHERE THE PHENYL OR BENCILO MAY BE REPLACED BY A GROUPS: C 1 C SUB, 6, ALCOXI C 1 - C 6, HALO, NITRO, AMINO OR TRIPLUO ROMETILO, YR 2 IS RENT C 1 - C 6, TRIFLUOROMETILO OR PHENYL, WHICH CAN BE REPLACED BY ONE OR MORE THAN GROUPS: RENT C 1 - C 6, ALCOXI C 1 - C SU B, 6, HALO, NITRO, AMINO OR TRIFLUOROMETILO, ASY AS AN INTERMEDIARY PREPARATION PROCEDURE I.
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机译:本发明涉及一种用于制备萘啶酮及其衍生物的羧酸的方法,该方法使用式I和式IV的侧链中间体,其中R 1为苯甲环,而苯基或苯甲环可以由以下基团取代:C 1 C取代基,6,ALCOXI C 1-C 6,卤素,硝基,氨基或三氟甲烷,YR 2出租C 1-C 6,三氟甲氧基或苯基,可以用一个或多个组代替:出租C 1-C 6 ,作为中间制备程序的ACOXI C 1-C SU B,6,晕,硝基,氨基或三氟甲磺酸,ASY。
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