首页> 外国专利> PHARMACEUTICAL COMPRISING (S)-4-AMINO-5-CHLORO-2-METHOXY-N-1-1-(2-TETRAHYDROFURYLCARBONYL)-4-PIPERIDINYLMETHYL-4-PIPERIDINYLBENZAMIDE

PHARMACEUTICAL COMPRISING (S)-4-AMINO-5-CHLORO-2-METHOXY-N-1-1-(2-TETRAHYDROFURYLCARBONYL)-4-PIPERIDINYLMETHYL-4-PIPERIDINYLBENZAMIDE

机译:包含(S)-4-氨基5-氯-2-甲氧基-N- [1- [1-(2-四氢呋喃基羰基)-4-哌啶基亚甲基乙基] -4-哌啶基]苯甲酰胺的药物

摘要

PROBLEM TO BE SOLVED: To obtain a pharmaceutical comprising a compound capable of strongly acting on a serotonin 4 receptor, extremely scarcely having an effect on the heart, without having a centric side effect caused by a dopamine D2 receptor, and useful as an enteric movement accelerating agent or an enteric function improving agent.;SOLUTION: This pharmaceutical comprises (S)-4-amino-5-chloro-2-methoxy-N-[1-[1-(2-tetrahydrofurylcarbonyl)-4-piperidinylmethyl]-4-piperidinyl]benzamide expressed by formula (I), its pharmaceutically acceptable acid addition salt, and a hydrate thereof.;COPYRIGHT: (C)2005,JPO&NCIPI
机译:要解决的问题:获得包含能够强烈作用于5-羟色胺4受体的化合物的药物,该化合物几乎对心脏几乎没有影响,而没有多巴胺D 2 引起的中枢性副作用;并可用作肠运动促进剂或肠功能改善剂。;解决方案:该药物包含(S)-4-氨基-5-氯-2-甲氧基-N- [1- [1-(2-由式(I)表示的四氢呋喃基羰基)-4-哌啶基甲基] -4-哌啶基]苯甲酰胺,其药学上可接受的酸加成盐及其水合物。;版权所有:(C)2005,JPO&NCIPI

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