首页> 外国专利> ESTERS OF L-CARNITINE OR ALKANOYL L-CARNITINE FOR USE AS CATIONIC LIPIDS FOR INTRA-CELLULAR ADMINISTRATION OF THERAPEUTIC SUBSTANCES

ESTERS OF L-CARNITINE OR ALKANOYL L-CARNITINE FOR USE AS CATIONIC LIPIDS FOR INTRA-CELLULAR ADMINISTRATION OF THERAPEUTIC SUBSTANCES

机译:左旋肉碱或烷基左旋肉碱的酯,用作治疗性药物细胞内给药的阳离子脂质

摘要

The use of esters of L-carnitine and alkanoyl L-carnitines as cationic lipids for the intracellular delivery of pharmacologically active compounds is described. The esters according to the invention have general formula (II) CHEM wherein the R groups are as defined in the description.
机译:描述了L-肉碱和烷酰基L-肉碱的酯作为阳离子脂质用于药理活性化合物的细胞内递送的用途。根据本发明的酯具有通式(II),其中R基团如说明书中所定义。

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