首页> 外国专利> COMBINATION PRODUCT COMPRISING AN ANTAGONIST OR INVERSE AGONIST OF HISTAMINE RECEPTOR HSB3 /SBAND AN ANTIPSYCHOTIC OR ANTIDEPRESSANT AGENT, AND USE THEREOF FOR THE PREPARATIONOF A MEDICAMENT THAT PREVENTS THE ADVERSE EFFECTS OF PSYCHOTROPIC DRUGS

COMBINATION PRODUCT COMPRISING AN ANTAGONIST OR INVERSE AGONIST OF HISTAMINE RECEPTOR HSB3 /SBAND AN ANTIPSYCHOTIC OR ANTIDEPRESSANT AGENT, AND USE THEREOF FOR THE PREPARATIONOF A MEDICAMENT THAT PREVENTS THE ADVERSE EFFECTS OF PSYCHOTROPIC DRUGS

机译:组合产品,其包含组胺受体H 3 的拮抗剂或逆激动剂和抗精神病药或抗抑郁药,并用于制备预防精神病药物不良作用的药物

摘要

A medicament comprising, in a pharmaceutically acceptable carrier, an anti-psychotic drug or an antidepressant (A), having only an adverse effect of body weight gain or sedation and an H3 receptor H3 receptor antagonist and / or inverse agonist (B) histamine, said histamine H3 receptor antagonist and / or inverse agonist being present in a therapeutically effective amount to achieve at least one of the following three effects: suppressing or at least limiting the adverse effect of taking weight, suppression or limitation of the adverse effect on alertness, epilepsy / seizures, increased pro-cognitive effect of treatment. Use of such an antagonist or inverse agonist for the preparation of a medicament for providing at least one of said three effects in a patient treated with such an antipsychotic or antidepressant.
机译:在药物可接受的载体中包含仅对体重增加或镇静有不良影响的抗精神病药或抗抑郁药(A)和H3受体,H3受体拮抗剂和/或反向激动剂(B)组胺,所述组胺H3受体拮抗剂和/或反向激动剂以治疗有效量存在,以实现以下三种作用中的至少一种:抑制或至少限制体重减轻的不利影响,抑制或限制对机敏性的不利影响,癫痫/癫痫发作,增加认知治疗的作用。所述拮抗剂或反向激动剂在制备药物中的用途,所述药物用于在用所述抗精神病药或抗抑郁药治疗的患者中提供所述三种作用中的至少一种。

著录项

  • 公开/公告号CA2530381A1

    专利类型

  • 公开/公告日2005-01-06

    原文格式PDF

  • 申请/专利权人 BIOPROJET;

    申请/专利号CA20042530381

  • 申请日2004-06-25

  • 分类号A61K31/551;A61K31/137;A61K31/40;A61K31/4025;A61K31/4412;A61K31/496;A61K31/513;A61K31/55;A61K31/554;A61P25/18;A61P25/24;

  • 国家 CA

  • 入库时间 2022-08-21 22:14:00

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