首页> 外国专利> PROCESS FOR PREPARATION OF ALPHA-HYDROXY-BENZENEACETIC ACID DERIVATIVES, AND PROCESS FOR PREPARATION OF COMPOUND HAVING TWO 5-MEMBERED LACTONE RINGS FUSED TO CENTRAL CYCLOHEXA-1,4-DIENE NUCLEUS USING THE SAME

PROCESS FOR PREPARATION OF ALPHA-HYDROXY-BENZENEACETIC ACID DERIVATIVES, AND PROCESS FOR PREPARATION OF COMPOUND HAVING TWO 5-MEMBERED LACTONE RINGS FUSED TO CENTRAL CYCLOHEXA-1,4-DIENE NUCLEUS USING THE SAME

机译:制备α-羟基-苯甲基乙酸衍生物的方法,以及使用相同的方法将具有两个5元内酯环的化合物融合到中央环己-1,4-二烯核中的方法

摘要

The invention cyclohexadiene-1, 4-diene-5 to the matrix in two essential raw materials for the production of compounds with a ring lock tonring alpha of formula - provides a process for the production of hydroxy-benzene acetic acid derivative. According to the method of the present invention, using a highly toxic substance, or without toxic substances it is not by-product can be easily produced the above compound in high purity and yield.; Wherein A, D 1 and R 1 are as defined in the specification.
机译:本发明以环己二烯-1、4-二烯-5为基质,在两种基本原料中生产具有式α的锁环的化合物-提供了一种生产羟基-苯乙酸衍生物的方法。根据本发明的方法,使用高毒性物质,或者不使用无毒物质,就可以容易地以高纯度和高收率生产上述化合物。其中,A,D 1 和R 1 如规范中所定义。

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