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therapeutic quassinoid preparations with anticancer, antiviral and herbistatischer effect

机译:具有抗癌,抗病毒和除草作用的治疗类quasinoid制剂

摘要

The present invention includes purified and isolated quassinoids and synthetically derived quassinoid analogs based on a picrasane carbon skeleton. Novel sidechains at C-15 incorporating water solubilizing agents such as glycine are discussed. Therapeutic methods taking advantage of anticancer, antiviral, and herbistatic properties of these quassinoids are disclosed, including use against solid tumors and human immunodeficiency virus infected cells. IMAGE
机译:本发明包括纯化的和分离的类胡萝卜素和基于异戊烷碳骨架的合成衍生的类胡萝卜素类似物。讨论了在C-15上加入水溶性试剂(如甘氨酸)的新型侧链。公开了利用这些类胡萝卜素的抗癌,抗病毒和除草特性的治疗方法,包括针对实体瘤和人类免疫缺陷病毒感染的细胞的用途。 <图像>

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