首页> 外国专利> USE OF GLUCOCORTICOID RECEPTOR MODULATORS AND GLUCOCORTICOID RECEPTOR AGONISTS FOR PREPARING MEDICAMENTS

USE OF GLUCOCORTICOID RECEPTOR MODULATORS AND GLUCOCORTICOID RECEPTOR AGONISTS FOR PREPARING MEDICAMENTS

机译:使用糖皮质激素受体调节剂和糖皮质激素受体激动剂制备药物

摘要

The present invention provides non-steroidal compounds of formula (I) which are selective modulators (i.e., agonists and antagonists) of a steroid receptor, specifically, the glucocorticoid receptor for the manufacture of a medicament for the treatment inflammation such as arthritis, asthma, rhinitis and immunomodulation in mammals and for reducing unwanted side effects using said treatment.
机译:本发明提供了式(I)的非甾体化合物,其为甾体受体,特别是糖皮质激素受体的选择性调节剂(即激动剂和拮抗剂),用于制备用于治疗炎症的药物,所述药物例如关节炎,哮喘,哺乳动物的鼻炎和免疫调节,以及使用所述治疗减少不必要的副作用。

著录项

  • 公开/公告号EA007483B1

    专利类型

  • 公开/公告日2006-10-27

    原文格式PDF

  • 申请/专利权人 PFIZER PRODUCTS INC.;

    申请/专利号EA20040000337

  • 申请日2000-03-27

  • 分类号C07C35/42;C07D295/12;A61K31/05;A61K31/122;A61K31/27;A61K31/275;A61K31/325;A61K31/40;A61K31/4164;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4965;A61K31/5375;A61P3/04;A61P3/10;A61P11/06;A61P19/02;A61P25/22;A61P25/24;A61P25/28;A61P27/16;A61P29;A61P37/02;A61P43;C07C49/675;C07C49/737;C07C49/747;C07C49/755;C07C49/757;C07C65/17;C07C69;C07C215/50;C07C215/74;C07C225/22;C07C233/58;C07C235/48;C07C235/66;C07C247/24;C07C251/44;C07C251/52;C07C251/60;C07C255/53;C07C255/54;C07C271/10;C07C271/44;C07C271/52;C07C281/04;C07C307/02;C07C309/65;C07C309/66;C07C309/73;C07C311/04;C07C311/08;C07C311/51;C07C317/18;C07C333/04;C07D207/09;C07D211/46;C07D213/22;C07D213/30;C07D213/40;C07D213/75;C07D231/40;C07D231/56;C07D233/61;C07D239/34;C07D241/12;C07D241/18;C07D241/20;C07D249/08;C07D249/14;C07D257/04;C07D271/06;C07D271/07;C07D277/24;C07D277/28;C07D277/56;C07D295/092;C07D295/13;C07D295/185;C07D295/205;C07D303/14;C07D317/36;C07D333/16;C07D413/04;C07D455/06;

  • 国家 EA

  • 入库时间 2022-08-21 21:39:38

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