首页> 外国专利> QUINOLINONE/BENZOXAZINONE DERIVATIVES AND USES THEREOF , PROCESSES FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND USES THEREOF IN THE PREPARATION OF MEDICAMENTS FOR TREATING OR PREVENTING A DISEASE STATE THAT IS ALLEVIATED BY 5HT6 AGONIST

QUINOLINONE/BENZOXAZINONE DERIVATIVES AND USES THEREOF , PROCESSES FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND USES THEREOF IN THE PREPARATION OF MEDICAMENTS FOR TREATING OR PREVENTING A DISEASE STATE THAT IS ALLEVIATED BY 5HT6 AGONIST

机译:喹诺酮/苯并恶嗪酮衍生物及其用途,其制备方法,包含它们的药物组合物及其在制备治疗或预防5HT6激动剂所致疾病的药物中的用途

摘要

The invention provides compounds of the formula: (I) and pharmaceutically acceptable salts or prodrugs thereof, wherein m, p, q, r, A, E, X, Y, R1, R4, R5, R6, R7, R8, R9 and are as defined herein. The invention also provides methods for preparing, compositions comprising, and methods for using compounds of formula I.
机译:本发明提供下式的化合物:(I)及其药学上可接受的盐或前药,其中m,p,q,r,A,E,X,Y,R1,R4,R5,R6,R7,R8,R9和如本文所定义。本发明还提供了制备式I的方法,包含式I的化合物的方法以及使用式I的化合物的方法。

著录项

  • 公开/公告号IL170439A

    专利类型

  • 公开/公告日2006-02-21

    原文格式PDF

  • 申请/专利权人 F. HOFFMANN-LA ROCHE AG;

    申请/专利号IL170439

  • 发明设计人

    申请日2005-08-22

  • 分类号

  • 国家 IL

  • 入库时间 2022-08-21 21:39:11

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