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A PROCESS FOR PREPARATION OF DOSAGE FORMULATION FOR ORAL ADMINISTRATION OF COX-2 INHIBITORS

机译:一种用于口服COX-2抑制剂的制剂的制备方法

摘要

The present invention describes a process of preparation pharmaceutical compositions for oral administration comprising of COX-2 inhibitors and wetting agent for improving dissolution and bioavailability of COX-2 inhibitors. In the present invention COX-2 inhibitor is in micronized form which helps in improving dissolution of poorly water soluble COX-2 inhibitors. The process of manufacturing of such pharmaceutical composition is also disclosed in the present invention. Drawing: NIL Total Pages: 22 Fig. Nil
机译:本发明描述了制备用于口服的药物组合物的方法包含COX-2抑制剂和湿润剂的药物给药,可改善药物的溶解度和生物利用度COX-2抑制剂。在本发明中,COX-2抑制剂为微粉化形式,有助于改善水溶性差的COX-2抑制剂的溶解。这种药物的制造过程本发明还公开了组合物。 绘图:NIL总页数:22图无

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