As an activator of melamycin m3 and / or M4 receptor

摘要

It is an oxopiridina derivative of the first equation, n is 1; RA, RA ',RB and rb'son h, cicoal quilo, etc.; R1 is asphalt or cyclopropyl; R2 is heterogeneous; R3 is halogen, asphalt, NO2, etc.; R5 is asphalt or cyclopropyl; R4 is a set of selected formulas.(b) And (c),a. Finally, it is changed to oxo group, or mono - or aggregate - or replaced by arilo group or heteromorphic group; P is 0, 1, 2 or 3; m is 0, 1 or 2; X is n (R10) link - or C (R6) (R7) - contact point;R6 is h, halogen, etc.; R7 is halogen, tar, etc.; R10 is cyclopropyl, arilo, etc. 1 - [4-1-1 - [4-1 - [4-1-1-1-phenol, including (a) cyclohexane, among others. A drug synthesis and preparation procedure was also mentioned. These compounds can be used to treat obesity, diabetes, sexual dysfunction and so on.