首页> 外国专利> n - idrossiammidi - substituted tricyclic groups as inhibitors of histone deacelitasi, their preparation and use in pharmaceutical formulations

n - idrossiammidi - substituted tricyclic groups as inhibitors of histone deacelitasi, their preparation and use in pharmaceutical formulations

机译:n-Idrossiammidi-取代的三环基团作为组蛋白去甲斑的抑制剂,其制备方法和在药物制剂中的用途

摘要

New N-hydroxyamides of n-alkyl carboxylic acids omega substituted with suitable tricyclic systems characterised by a central 7-membered ring, having activity as inhibitors of histone deacetylase (HDAC).
机译:由合适的三环系统取代的新型正构烷基ω-脂肪酸的N-羟酰胺,其特征在于中心的7元环,具有作为组蛋白脱乙酰基酶(HDAC)抑制剂的活性。

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