首页> 外国专利> N-(3-(IMIDAZO 1,5-APYRIMIDIN-4-YL)PHENYL-SULFONAMIDES AND N-3-(IMIDAZO1,5-APYRIMIDIN-4-YL)-PHENYL-CARBOXAMIDES AND THEIR USE AS GABAA RECEPTOR MODULATORS

N-(3-(IMIDAZO 1,5-APYRIMIDIN-4-YL)PHENYL-SULFONAMIDES AND N-3-(IMIDAZO1,5-APYRIMIDIN-4-YL)-PHENYL-CARBOXAMIDES AND THEIR USE AS GABAA RECEPTOR MODULATORS

机译:N-(3-(咪唑并[1,5-A]吡喃基-4-基]苯基]-磺酰胺和N- [3-(咪唑并[1,5-A]吡喃基-4-基]-苯基]-羧酰胺及其作为GABAA受体调节剂的用途

摘要

The present invention relates to compounds of formula I wherein R1, R2, R3 and X are as defined in the claims. The compounds have specific affinity for the GABAA receptor and are therefore useful in the treatment and prevention of diseases modulated by the 1 and 2-GABAA receptors.
机译:本发明涉及式I化合物,其中R 1,R 2,R 3和X如权利要求所定义。该化合物对GABAA受体具有特定的亲和力,因此可用于治疗和预防由1和2-GABAA受体调节的疾病。

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