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INHALATION MEDICINES CONTAINING A NEW ANTICHOLINERGIC MEDICINE IN COMBINATION WITH CORTICOSTEROIDS AND BETAMETHYMETICS

机译:包含抗肠线虫药物和糖皮质激素和双药合用的新型吸入药物

摘要

An inhalable medicament (A) comprises a combination of 6beta,7beta-epoxy-3beta-hydroxy-8-methyl-1alphaH,5alpha-H-tropanium salt 2,2-diphenylpropionate ester anticholinergic agent(s) (I) and EFGR kinase inhibitor(s) (II), optionally together with auxiliaries. An inhalable medicament (A) comprises a combination of tropane derivative anticholinergic agent(s) of formula (I), corticosteroid(s) (II) and beta-mimetic agent(s) (III) (optionally in the form of enantiomers, enantiomer mixtures or racemates, or solvates or hydrates), optionally together with pharmaceutical auxiliaries. X- = monovalent anion, preferably chloride, bromide, iodide, sulfate, phosphate, methanesulfonate, nitrate, maleate, acetate, citrate, fumarate, tartrate, oxalate, succinate, benzoate or p-toluenesulfonate.
机译:可吸入药物(A)包含6beta,7beta-环氧-3beta-羟基-8-甲基-1alphaH,5alpha-H-托pan盐2,2-二苯丙酸酯抗胆碱药(I)和EFGR激酶抑制剂的组合(s)(II),可选配助剂。可吸入药物(A)包含式(I)的托烷衍生物抗胆碱能药,皮质类固醇(II)和β-模拟药(III)的组合(任选地以对映异构体,对映异构体的形式)混合物或外消旋物,或溶剂化物或水合物),以及药物助剂。 X-=一价阴离子,优选氯离子,溴离子,碘离子,硫酸根,磷酸根,甲磺酸根,硝酸根,马来酸根,乙酸根,柠檬酸根,富马酸根,酒石酸根,草酸根,琥珀酸根,苯甲酸根或对甲苯磺酸根。

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