首页> 外国专利> Crystals of E-2-methoxy-N- (3- {4- 3-methyl-4- (6-methyl-pyridin-3-yloxy) -phenylamino -quinazolin-6-yl} -allyl) -acetamide

Crystals of E-2-methoxy-N- (3- {4- 3-methyl-4- (6-methyl-pyridin-3-yloxy) -phenylamino -quinazolin-6-yl} -allyl) -acetamide

机译:E-2-甲氧基-N-(3- {4- [3-甲基-4-(6-甲基-吡啶-3-基氧基)-苯氨基]-喹唑啉-6-基}-烯丙基)-乙酰胺的晶体

摘要

Crystal forms of E-2-Methoxy-N-(3-{4-[3-methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide. A crystal form is useful in the synthesis of salts and complexes of E-2-Methoxy-N-(3-{4-[3-methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide. A crystal form also improves stability of tabletted or capsuled E-2-Methoxy-N-(3-{4-[3-methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide as a drug product.
机译:E-2-甲氧基-N-(3- {4- [3-甲基-4-(6-甲基-吡啶-3-基氧基)-苯氨基]-喹唑啉-6-基}-烯丙基)-乙酰胺的晶体形式。晶体形式可用于合成E-2-甲氧基-N-(3- {4- [3-甲基-4-(6-甲基-吡啶-3-基氧基)-苯基氨基]-喹唑啉的盐和配合物-6-基}-烯丙基)-乙酰胺。晶型还改善了片剂化或胶囊化的E-2-甲氧基-N-(3- {4- [3-甲基-4-(6-甲基-吡啶-3-基氧基)-苯基氨基]-喹唑啉-6- yl}-烯丙基)-乙酰胺为药物产品。

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