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Pirazolopirimidinas

机译:皮拉佐皮里米吉纳

摘要

Pirazolopirimidinas of Formula 1, in which the symbols have the following Meanings: R1 is Hydrogen, alkyl substituted alquenilo Case since, in case in case alquinilo substituted cycloalkyl substituted cycloalkyl substituted in case if necessary, substitute In case heterociclilo Gone or replaced, Hydroxy, alkoxy substituted amino, if given,Alquilamino in case in case dialquilamino replaced or substituted alkyl; R2 is Hydrogen or; or R1 and R2 mean along with the nitrogen Atom, which are linked to a Heterocyclic ring, IF R3 is replaced; if given aryl substituted, and In case rociclilo substituted alkyl substituted in given case.Alquenilo in case in case alquinilo substituted cycloalkyl substituted, IF replaced, cicloalquenilo in case in case aralquilo substituted Halogen substituted amino Group in a given case (C1 - alkoxy substituted, - 8) in the case Alquiltio substituted C1 - 8 - If replaced, ariloxi c6-10 if replaced,Ariltio - C6 - 10 in case in case heterocicliloxi substituted aryl substituted, - C6 - 10 - alcoxic1 - 4 in case ariloc6 substituted, - 10 - in case Alquiltio c1-4 alkoxy substituted, heterociclil - C1 - 4 in case replaced, heterociclil - Alquiltio - C1 - 4 in case substituted 0R8 (C, S) C (or SR8) or C (S) conr6r7 SR8 R4 R5 means; means; h, halogen, alkyl substitutedIn case, cycloalkyl substituted by Halogen, halogen, in case the Dodo, or c1-4 alkyl, or s (o) 0 - 2 - 4 - C1 - alkyl; X is halogeno, cyano substituted alkyl, Hydroxy, in case halogenoalquilo c1-3, alkoxy substituted phenyl in given case. Replaced in case, Alquiltio substitute Gone in a given case.In case alquilsulfinil substituted or replaced in case alquilsulfonilo R6 H means; for example, a cation substituted Ammonium ion in a given case by alkyl or arylalkyl substituted alkyl, IF alquenilo replaced in case, alquinilo replaced if In case cicloalquenilo cycloalkyl substituted and replaced if necessary.Aryl substituted arylalkyl substituted in given case and if necessary; R7 means cor8, S (OR) 1 - 2r8, cyano, coor8, (R8) 2, May be the remains of a Ring heterocycle R8, with 5 or 6 members fully or partially saturated unsaturated if replaced, identical or different, cont So, in case 1 or up to three additional heteroatoms selected from Atoms n, s and / or orWithout Oxygen Atoms can be contiguous; R8 are independently h, alkyl substituted halogenoalquilo Case since, in case alquenilo replaced, in case in case alquinilo substituted cycloalkyl substituted, IF replaced, ciclaolqueni In case it replaced,In case aralquilo substituted aryl or substituted if necessary; or two remains R8 form a cycle C3 - 6, which is partially saturated or unsaturated, and contains, in case, 1 or 2 Atoms n, s or without additional Oxygen Atoms can be contiguous or R6 and; R8 form In conjunction with the groups co n - or N - S (o) 1 - 2, on which are linked.A cycle with 4 - 8 members that may contain one or more heteroatoms from the group consisting of oxygen and / or Sulphur, nitrogen, and Oxygen Atoms to be contiguous; as well as als salts with Agrochemical Business of the same.
机译:式1的Pirazolopirimidinas,其中的符号具有以下含义:R1是氢,烷基取代的alquenilo情况,因为在必要的情况下,如果情况下被alquinilo取代的环烷基取代的环烷基取代,则在情况下被取代,在杂环基被取代或被取代时,羟基,烷氧基取代的氨基(如果有的话),如果用dialquilamino取代或取代的烷基,则Alquilamino; R 2为氢或; R 1和R 2表示与杂环连接的氮原子,如果R 3被取代;如果给定的情况下是芳基取代的,在给定的情况下是rociclilo取代的烷基;在给定的情况下,alquelolo被卤素取代的氨基(C1-烷氧基取代, -8)如果Alquiltio取代了C1-8-如果被取代,则将ariloxi c6-10取代,如果是异环己烯基取代的芳基,则将Ariltio-C6-10取代了,-如果将ariloc6取代了芳基环烷基,将-C6-10-alcoxic1-4取代了,- 10-如果Alquiltio c1-4烷氧基被取代,杂基-C1-4被取代,杂基-Alquiltio-C1-4如果被取代0R8(C,S)C(或SR8)或C(S)conr6r7 SR8 R4 R5手段;手段; h,卤素,被烷基取代的情况,如果环烷基被卤素,卤素,如果渡渡鸟,或c 1-4烷基,或s(o)0 -2-4-C 1-烷基取代; X是卤代,氰基取代的烷基,羟基,在给定情况下,在卤代α1-3的情况下是烷氧基取代的苯基。如果替换,则在特定情况下用Alquiltio代替。如果用alquilsulfonilo R6 H表示,则用Alquilsulfinil取代或替换。例如,给定情况下被烷基或芳基烷基取代的烷基取代的阳离子铵离子,如果情况下被Alquenilo取代,则被Alquinilo取代;如果被Cicloalquenilo环烷基取代,则被Alquinilo取代;必要时被取代。 R7表示cor8,S(OR)1-2r8,氰基,coor8,(R8)2,可能是环杂环R8的残基,如果被取代,相同或不同,则5或6个成员完全或部分饱和,续,如果从原子n,s和/或无氧原子中选择1个或最多3个其他杂原子,则可以是连续的; R8独立地是h,烷基取代的卤代烷基,因为如果用alquenilo取代,如果用alquinilo取代的环烷基取代,如果用IF取代,ciclaolqueni。或两个残基R8形成部分饱和或不饱和的环C3-6,并且在1或2个原子n,s或不具有另外的氧原子的情况下可以是连续的或R6,并且; R8形式与连接在其上的基团co n-或N-S(o)1-2结合。一个具有4-8个成员的循环,这些成员可能包含一个或多个选自氧和/或的杂原子硫,氮和氧原子是连续的;以及与农用化学品业务相同的ALS盐。

著录项

  • 公开/公告号AR052913A1

    专利类型

  • 公开/公告日2007-04-11

    原文格式PDF

  • 申请/专利权人 BAYER CROPSCIENCE AG;

    申请/专利号AR2006P100581

  • 发明设计人

    申请日2006-02-17

  • 分类号C07D487/04;A01N43/90;C07D231/00;C07D239/00;C07D487/04;

  • 国家 AR

  • 入库时间 2022-08-21 20:59:39

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