首页> 外国专利> DIPEPTIDYL PEPTIDASE INHIBITING 7-(3-AMINO-4-ARYLBUTANOYL)TETRAHYDROIMIDAZO (1,2-A) PYRAZINE AND TETRAHYDROTRIAZOLO (4,3-A) PYRAZINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

DIPEPTIDYL PEPTIDASE INHIBITING 7-(3-AMINO-4-ARYLBUTANOYL)TETRAHYDROIMIDAZO (1,2-A) PYRAZINE AND TETRAHYDROTRIAZOLO (4,3-A) PYRAZINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

机译:抑制7-(3-氨基-4-芳基丁酰基)四氢咪达唑(1,2-A)吡嗪和四氢三唑(4,3-A)吡嗪衍生物和包含它们的药物组合物的二肽肽酶

摘要

The present invention is directed to pharmaceutical compositions comprising compounds which are inhibitors of the dipeptidyl peptidase-IV enzyme ("DP-IV inhibitors") and the use of these compositions in the treatment or prevention of diseases in which the dipeptidyl peptidase-IV enzyme is involved, such as diabetes and particularly type 2 diabetes.
机译:本发明涉及包含作为二肽基肽酶-IV酶的抑制剂的化合物(“ DP-IV抑制剂”)的药物组合物,以及这些组合物在治疗或预防其中二肽基肽酶-IV酶为疾病的疾病中的用途。涉及,例如糖尿病,尤其是2型糖尿病。

著录项

  • 公开/公告号IL159109B

    专利类型

  • 公开/公告日2007-06-03

    原文格式PDF

  • 申请/专利权人 MERCK SHARP & DOHME CORP.;

    申请/专利号IL159109

  • 发明设计人

    申请日2003-11-27

  • 分类号A61K31/498;A61K31/4985;A61K45/00;A61K45/06;A61P1/02;A61P1/04;A61P3/04;A61P3/06;A61P3/10;A61P5/06;A61P5/28;A61P5/50;A61P7/00;A61P9/08;A61P9/10;A61P9/12;A61P13/08;A61P13/12;A61P15/16;A61P19/10;A61P25/00;A61P25/28;A61P27/02;A61P31/18;A61P35/04;A61P37/02;A61P43/00;C07D487/04;

  • 国家 IL

  • 入库时间 2022-08-21 20:58:40

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号