首页> 外国专利> METHODS FOR THE DRUG PROPHYLAXIS OF POISONING BY CHOLINESTERASE INHIBITORS, AND ACTIVE INGREDIENTS AND MEDICAMENTS SUITABLE THEREFORE

METHODS FOR THE DRUG PROPHYLAXIS OF POISONING BY CHOLINESTERASE INHIBITORS, AND ACTIVE INGREDIENTS AND MEDICAMENTS SUITABLE THEREFORE

机译:胆碱酯酶抑制剂中毒的药物预防方法以及因此所需的活性成分和药物

摘要

Dialkylaminoalkylphenyl carbamate derivatives (I) are used to protect people from poisoning by cholinesterase inhibitors. Dialkylaminoalkylphenyl carbamate derivatives of formula (I) are used to protect humans from poisoning with cholinesterase inhibitors. R1 = H, 1-5C alkyl, cyclohexyl, allyl or benzyl; R2 = H, Me, Et or Pr; R3 = H or 1-5C alkyl; and R4, R5 = 1-5C alkyl. An Independent claim is also included for a medicament for preventing poisoning by cholinesterase inhibitors, comprising at least one compound (I) is free base or salt form and one or more parasympatholytic agents.
机译:二烷基氨基烷基苯基氨基甲酸酯衍生物(I)用于保护人们免受胆碱酯酶抑制剂的中毒。式(I)的二烷基氨基烷基苯基氨基甲酸酯衍生物用于保护人类免受胆碱酯酶抑制剂的中毒。 R1 = H,1-5C烷基,环己基,烯丙基或苄基; R 2 = H,Me,Et或Pr; R3 = H或1-5C烷基;和R4,R5 = 1-5C烷基。还包括用于预防胆碱酯酶抑制剂中毒的药物的独立权利要求,所述药物包含至少一种为游离碱或盐形式的化合物(I)和一种或多种副交感神经药。

著录项

  • 公开/公告号IL169687D0

    专利类型

  • 公开/公告日2007-07-04

    原文格式PDF

  • 申请/专利权人 LTS LOHMANN THERAPIE-SYSTEME AG;

    申请/专利号IL20050169687

  • 发明设计人

    申请日2005-07-14

  • 分类号A61K31/325;A61K31/46;C07C;

  • 国家 IL

  • 入库时间 2022-08-21 20:58:38

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