It refers to a kind of drug synthesis, including: (a) acid 1 - [4 - (2-azepan-1-il-etoxi) - bencil] - 2 - (4-hydroxifenil) - 3-met-1h-indol-5-ol acetic (acetic acid of bazedoxiphen) as a form of crystalline polymorphone, with a content of 0.1-30% by weight of preparation; (b) as the first filling / diluent of sugar, Microcrystalline cellulose, starch, etc., the content is 5-85% by formula weight; (c) the content of the second filling / diluent, such as lactose, is 5-85% by formula weight; (d) An antioxidant, such as acido ascorbico, with a content up to 15% by weight of the formula;(e) A sliding / decomposing agent, such as starch glycerin, containing between 0.01% and 10% by formula weight; F) lubricating oil, such as magnesium stearate, containing between 0.01% and 10% by formula weight. He also mentioned a procedure for preparing music. As a selective modulator of estrogen receptor, diacetate is very useful in the treatment of postmenopausal osteoporosis.
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