首页> 外国专利> AMIDES OF MONO AND BICARBOXYLIC ACIDS WITH AMINO ACIDS OR GLYCOSAMINES, SELECTIVELY ACTIVE ON THE CANNABINOID PERIPHERAL RECEPTOR

AMIDES OF MONO AND BICARBOXYLIC ACIDS WITH AMINO ACIDS OR GLYCOSAMINES, SELECTIVELY ACTIVE ON THE CANNABINOID PERIPHERAL RECEPTOR

机译:单价和双羧酸与氨基酸或糖胺的酰胺,对大麻素外围受体具有选择性活性

摘要

The present invention relates to amides offormula (I):wherein R1 is an optionally substituted linear or branchedhydrocarbon radical, or a group of formula (II) or (III):wherein R4 is an optionally substituted linear hydrocarbonradical, R7 is H or a linear or branched alkyl, and theresiduesare glycosaminic residues; a pharmaceutical compositioncomprising the amide; and a use of the amide as a CB2receptor modulator.
机译:本发明涉及甲酰胺公式(I):其中R1是任选取代的直链或支链烃基或式(II)或(III)的基团:其中R4为任选取代的直链烃R 7是氢或直链或支链烷基,并且残渣是糖胺残基;药物组合物包含酰胺;以及酰胺作为CB2的用途受体调节剂。

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