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EPIDURAL ADMINISTRATION OF THERAPEUTIC COMPOUND WITH SUSTAINED RATE OF RELEASE

机译:具有持续释放率的治疗化合物的硬膜外给药

摘要

PPROBLEM TO BE SOLVED: To provide sustained release delivery of a physiologically active therapeutic administered epidurally. PSOLUTION: A liposome preparation for treating the pain after surgery of a vertebrate animal or after delivery is epidurally administered as a single dose and comprises an analgetic compound or an anesthetic compound encapsulated within multi-vesicular liposomes, and the analgetic compound or the anesthetic compound is sustainedly released. PCOPYRIGHT: (C)2008,JPO&INPIT
机译:

要解决的问题:提供硬膜外给药的生理活性治疗剂的缓释递送。

解决方案:用于治疗脊椎动物手术后或分娩后疼痛的脂质体制剂以单剂量硬膜外给药,并且包含麻醉性化合物或封装在多囊脂质体内的麻醉剂,以及该麻醉性化合物或麻醉化合物持续释放。

版权:(C)2008,日本特许厅&INPIT

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