首页> 外国专利> 2, 8-DIMETHYL-5- 2- (6-METHYLPYRIDIN-3-YL) -ETHYL -2,3,4, 5-TETRAHYDRO- IH- PYRIDO 4, 3 -B INDOLE DIHYDROCHLORIDE (DIMEBON) FOR THE TREATMENT OF CHRONIC PAIN

2, 8-DIMETHYL-5- 2- (6-METHYLPYRIDIN-3-YL) -ETHYL -2,3,4, 5-TETRAHYDRO- IH- PYRIDO 4, 3 -B INDOLE DIHYDROCHLORIDE (DIMEBON) FOR THE TREATMENT OF CHRONIC PAIN

机译:2,8,8-二甲基-5- [2-(6-甲基吡啶-3-基)-乙基] -2,3,4,5-四氢-IH-吡咯烷[4,3 -B]吲哚二氯(DIMEBON)慢性疼痛的治疗

摘要

The present invention provides methods of treating chronic pain, in particular, neuropathic pain, chronic visceral pain, chronic inflammatory pain and pain resulting from fibromyalgia syndrome, in a subject by administering Dimebon™ antihistamine agent (DETCD) to the subject. The invention also provides methods of treating chronic pain in a subject by administering a combination of DETCD and one or more additional agents, such as an antidepressant agent, an anticonvulsant agent, an antiarrhythmic agent, an anesthetic agent, an NMDA antagonist, or a narcotic.
机译:本发明提供了通过将Dimebon TM抗组胺药(DETCD)施用于受试者来治疗受试者的慢性疼痛,特别是神经性疼痛,慢性内脏疼痛,慢性炎症性疼痛和由纤维肌痛综合征引起的疼痛的方法。本发明还提供了通过施用DETCD和一种或多种另外的药物例如抗抑郁药,抗惊厥药,抗心律不齐药,麻醉药,NMDA拮抗剂或麻醉药的组合来治疗受试者的慢性疼痛的方法。 。

著录项

  • 公开/公告号WO2008112238A1

    专利类型

  • 公开/公告日2008-09-18

    原文格式PDF

  • 申请/专利权人 GREY FOX LLC;HERLANDS LOUIS;

    申请/专利号WO2008US03246

  • 发明设计人 HERLANDS LOUIS;

    申请日2008-03-12

  • 分类号A61K31/437;A61P25/04;A61P25/06;A61P29;A61P29/02;A61P21;

  • 国家 WO

  • 入库时间 2022-08-21 19:57:13

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