首页> 外国专利> PYRAZOLO 1,5-A PYRIDINES COMPOUNDS HAVING CORTICOTROPIN-RELEASING FACTOR RECEPTOR ANTAGONISTIC ACTIVITY, SALTS THEREOF HYDRATES OF THE FOREGOING

PYRAZOLO 1,5-A PYRIDINES COMPOUNDS HAVING CORTICOTROPIN-RELEASING FACTOR RECEPTOR ANTAGONISTIC ACTIVITY, SALTS THEREOF HYDRATES OF THE FOREGOING

机译:具有释放促肾上腺皮质激素的因子受体拮抗活性的吡咯并[1,5-A]吡啶化合物,其盐类如前所述。

摘要

[wherein R1 represents methoxy, ethyl, methylthio, etc., R2, R3 and R4 each represent hydrogen, a halogen, etc., R5 and R6 each represent - X5-X6-X7 (wherein X5 represents a single bond or -CO-, X6 represents a single bond, NR3a, etc. and X7 and R3a each represent hydrogen, C1-10 alkyl, etc.), and Ar represents phenyl, pyridyl, etc.], salts thereof and hydrates of the foregoing.
机译:[其中R1代表甲氧基,乙基,甲硫基等,R2,R3和R4各自代表氢,卤素等,R5和R6各自代表-X5-X6-X7(其中X5代表单键或-CO- [式中,X 6表示单键,NR 3a等,X 7和R 3a分别表示氢,C 1-10烷基等),Ar表示苯基,吡啶基等。],其盐和它们的水合物。

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