首页> 外国专利> 5-HALO-TRYPTAMINE DERIVATIVES USED AS LIGANDS OF THE 5-HT 6? AND/OR 5-HT 7? SEROTONIN RECEPTORS

5-HALO-TRYPTAMINE DERIVATIVES USED AS LIGANDS OF THE 5-HT 6? AND/OR 5-HT 7? SEROTONIN RECEPTORS

机译:用作5-HT 6配体的5-卤代色胺衍生物吗?和/或5-HT 7?血清素受体

摘要

Compounds of Formula (I): (I); wherein: RSUB1 /SUBand RSUB2 /SUBeither the same or different, are H or linear or branched CSUB1/SUB-CSUB6 /SUBalkyl; RSUB3/SUB=linear or branched CSUB1/SUB-CSUB6 /SUBalkyl; RSUB4/SUB=halogen, and pharmaceutically acceptable salts thereof are useful as active ingredients in the preparation of medicaments used as ligands of the 5-HTSUB6 /SUBand/or 5-HTSUB7 /SUBserotoninergic receptors.
机译:式(I)的化合物:其中:R 1 和R 2 相同或不同,为H或直链或支链的C 1 -C 6 烷基; R 3 =直链或支链C 1 -C 6 烷基; R 4 =卤素及其药学上可接受的盐可用作活性成分,用于制备用作5-HT 6 和/或5-HT < SUB> 7 5-羟色胺能受体。

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