首页> 外国专利> A PHARMACEUTICAL COMPOSITION CONTAINING SUBSTITUTED BICYCLO 3.3.1 NONAN-2,4,9-TRIONES AS AN ACTIVE INGREDIENTS FOR PROPHYLACTIC AND/OR THERAPEUTIC TREATMENT OF NEOPLASTIC OR CANCEROUS DISEASE AND VIRAL DISEASES

A PHARMACEUTICAL COMPOSITION CONTAINING SUBSTITUTED BICYCLO 3.3.1 NONAN-2,4,9-TRIONES AS AN ACTIVE INGREDIENTS FOR PROPHYLACTIC AND/OR THERAPEUTIC TREATMENT OF NEOPLASTIC OR CANCEROUS DISEASE AND VIRAL DISEASES

机译:包含取代的双环[3.3.1] NONAN-2,4,9-三酮类药物的药物组合物,可作为活性成分治疗坏死性或癌性疾病和病毒性疾病的预防性和/或治疗性药物

摘要

The invention relates to the use of substituted bicyclo [3.3.1] nonan-2,4,9-triones, especially clusianon and clusianon derivatives, as pharmaceutical active ingredients or medicamentous active ingredients, especially for producing medicaments for the prophylactic and/or therapeutic (curative) treatment of tumour or cancer diseases, and of viral diseases. The above-mentioned compounds can be used in cytostatic agents and antiviral agents (virostatic agents). They are especially used as inhibitors of topoisomerases and telomerases and as regulators during the MAP kinase signal transduction and can thus intervene on a cellular scale in the mechanism for multiplication of tumour or cancer cells and viruses.
机译:本发明涉及取代的双环[3.3.1]壬二-2,4,9-三酮,特别是clusianon和clusianon衍生物作为药物活性成分或药物活性成分的用途,特别是用于生产预防和/或治疗药物(治愈)治疗肿瘤或癌症疾病以及病毒性疾病。上述化合物可以用于细胞抑制剂和抗病毒剂(抗病毒剂)中。它们特别用作拓扑异构酶和端粒酶的抑制剂,以及在MAP激酶信号转导过程中的调节剂,因此可以在细胞规模上干预肿瘤或癌细胞和病毒的增殖机制。

著录项

  • 公开/公告号IN239087B

    专利类型

  • 公开/公告日2010-03-12

    原文格式PDF

  • 申请/专利权人

    申请/专利号IN337/MUMNP/2004

  • 申请日2004-06-15

  • 分类号A61K35/64;A61K31/12;

  • 国家 IN

  • 入库时间 2022-08-21 18:45:56

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