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DOUBLE-LAYERED ZALEPLON-CONTAINED TABLET

机译:双层双层扎普龙含片剂

摘要

PURPOSE: A double-layered tablet containing zaleplon is provided to improve stability of medicinal use and convenience and improve sleeping quality. CONSTITUTION: A double-layered zaleplon-containing tablet contains immediate release layer and sustained release layer. The tablet is produced by stirring 0.1N of hydrochloric acid buffer and pH 6.8 of phosphoric acid buffer at 50-200rpm. The immediate release layer contains zaleplon, lactose, maltose, microcrystalline cellulose, Sodiumlauryl sulfate and at least one additive. The sustained release layer contains zaleplon, maltose, microcrystalline cellulose, polymer and at least one additive. The additive is disintegrant, glidant, or lubricant.
机译:目的:提供一种含扎来普隆的双层片剂,以提高药物使用的稳定性和便利性,并改善睡眠质量。组成:含扎来普隆的双层片剂包含立即释放层和持续释放层。通过在50-200rpm下搅拌0.1N盐酸缓冲液和pH 6.8磷酸缓冲液来生产片剂。速释层包含扎来普隆,乳糖,麦芽糖,微晶纤维素,月桂基硫酸钠和至少一种添加剂。持续释放层包含扎来普隆,麦芽糖,微晶纤维素,聚合物和至少一种添加剂。添加剂是崩解剂,助流剂或润滑剂。

著录项

  • 公开/公告号KR20100020893A

    专利类型

  • 公开/公告日2010-02-23

    原文格式PDF

  • 申请/专利权人 ORIENT PHARMA CO. LTD.;

    申请/专利号KR20090019173

  • 发明设计人 WEN TING KE;TSE CHING LIN;

    申请日2009-03-06

  • 分类号A61K9/22;A61P25;A61K31/519;A61K47/38;

  • 国家 KR

  • 入库时间 2022-08-21 18:33:15

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