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Preventive and/or remedy for lower urinary tract diseases containing EP4 agonist

机译:含有EP 4 激动剂的下尿路疾病的预防和/或治疗

摘要

(1) A preventive and/or a remedy for lower urinary tract diseases such as inflammation in the lower urinary tract, cystitis (interstitial cystitis, etc.) and urethritis; (2) an agent for improving bladder compliance and/or bladder capacity; and (3) an agent for protecting bladder mucosa and/or bladder epithelial cells and/or promoting the regeneration thereof; each containing an EP4 agonist.;An EP4 agonist is useful in ameliorating symptoms of lower urinary tract diseases such as (1) frequent urination, (2) urgency of urination, (3) pain in the reproductive organs and/or lower urinary tract (for example, bladder pain, urinary tract pain, vulvar pain, vaginal pain, scrotal pain, perineal pain, pelvic pain, etc.) and/or (4) discomfort in the reproductive organs and/or lower urinary tract. Among all, a selective EP4 agonist is useful as a preventive and/or remedy for lower urinary tract diseases having no side effect.
机译:(1)对下尿路疾病的预防和/或治疗,例如下尿路炎症,膀胱炎(间质性膀胱炎等)和尿道炎; (2)用于改善膀胱顺应性和/或膀胱容量的试剂; (3)保护膀胱粘膜和/或膀胱上皮细胞和/或促进其再生的药剂。每种都包含EP 4 激动剂; EP 4 激动剂可用于缓解下尿路疾病的症状,例如(1)频繁排尿,(2)排尿急迫,(3)生殖器官和/或下尿路疼痛(例如,膀胱疼痛,尿路疼痛,外阴痛,阴道疼痛,阴囊痛,会阴痛,骨盆痛等)和/或(4)生殖器官和/或下尿路不适。其中,选择性的EP 4 激动剂可用作无副作用的下尿路疾病的预防和/或治疗方法。

著录项

  • 公开/公告号US7858610B2

    专利类型

  • 公开/公告日2010-12-28

    原文格式PDF

  • 申请/专利权人 HIROKI OKADA;TAKAYUKI MARUYAMA;

    申请/专利号US20050660043

  • 发明设计人 HIROKI OKADA;TAKAYUKI MARUYAMA;

    申请日2005-08-09

  • 分类号A61K31/54;A61K31/535;

  • 国家 US

  • 入库时间 2022-08-21 18:08:04

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